SAHORES, ANA; GONZÁLEZ, ANGELA RODRÍGUEZ; YANEFF, AGUSTÍN; MAY, MARÍA; GÓMEZ, NATALIA; MONCZOR, FEDERICO; FERNÁNDEZ, NATALIA; DAVIO, CARLOS; SHAYO, CARINA

Ceefourin-1, a MRP4/ABCC4 inhibitor, induces apoptosis in AML cells enhanced by histamine

BIOCHIMICA ET BIOPHYSICA ACTA-GENERAL SUBJECTS; Año: 2023 vol. 1867

ZÁRATE, LORENA V.; MIRET, NOELIA V.; NICOLA CANDIA, ALEJANDRO J.; ZAPPIA, C. DANIEL; PONTILLO, CAROLINA A.; CHIAPPINI, FLORENCIA A.; MONCZOR, FEDERICO; CANDOLFI, MARIANELA; RANDI, ANDREA S.

Breast cancer progression and kynurenine pathway enzymes are induced by hexachlorobenzene exposure in a Her2-positive model

FOOD AND CHEMICAL TOXICOLOGY; Año: 2023 vol. 177

GRANJA-GALEANO, GINA; DOMINGUEZ-RUBIO, ANA PAULA; ZAPPIA, C. DANIEL; WOLFSON, MANUEL; SANZ-BLASCO, SARA; AISEMBERG, JULIETA; ZORRILLA-ZUBILETE, MARIA; FERNANDEZ, NATALIA; FRANCHI, ANA; FITZSIMONS, CARLOS P.; MONCZOR, FEDERICO

CB1 receptor expression and signaling are required for dexamethasone-induced aversive memory consolidation

NEUROPHARMACOLOGY; Año: 2023 vol. 239

ECHEVERRÍA, EMILIANA; RIPOLL, SONIA; FABIÁN, LUCAS; SHAYO, CARINA; MONCZOR, FEDERICO; FERNÁNDEZ, NATALIA C.

Novel inhibitors of phosphorylation independent activity of GRK2 modulate cAMP signaling

Pharmacology Research and Perspectives; Año: 2022 vol. 10

MONCZOR, FEDERICO; GENARO, ANA

South American special issue: Editorial

Pharmacology Research and Perspectives; Año: 2021 vol. 9

BURGHI, VALERIA; ECHEVERRÍA, EMILIANA B.; ZAPPIA, CARLOS D.; DÍAZ NEBREDA, ANTONELA; RIPOLL, SONIA; GÓMEZ, NATALIA; SHAYO, CARINA; DAVIO, CARLOS A.; MONCZOR, FEDERICO; FERNÁNDEZ, NATALIA C.

Biased agonism at histamine H1 receptor: Desensitization, internalization and MAPK activation triggered by antihistamines

EUROPEAN JOURNAL OF PHARMACOLOGY; Año: 2021 vol. 896

RODRÍGUEZ GONZÁLEZ, ANGELA; SAHORES, ANA; DÍAZ-NEBREDA, ANTONELA; YANEFF, AGUSTÍN; DI SIERVI, NICOLÁS; GÓMEZ, NATALIA; MONCZOR, FEDERICO; FERNÁNDEZ, NATALIA; DAVIO, CARLOS; SHAYO, CARINA

MRP4/ABCC4 expression is regulated by histamine in acute myeloid leukemia cells, determining cAMP efflux

FEBS JOURNAL; Año: 2021

ZAPPIA, C. DANIEL; TORRALBA-AGU, VALERIA; ECHEVERRIA, EMILIANA; FITZSIMONS, CARLOS P.; FERNANDEZ, NATALIA; MONCZOR, FEDERICO

Antihistamines Potentiate Dexamethasone Anti-Inflammatory Effects. Impact on Glucocorticoid Receptor-Mediated Expression of Inflammation-Related Genes

Cells; Año: 2021 vol. 10

MIRET, NOELIA; ZAPPIA, C. DANIEL; ALTAMIRANO, GABRIELA; PONTILLO, CAROLINA; ZÁRATE, LORENA; GÓMEZ, AYELÉN; LASAGNA, MARIANELA; COCCA, CLAUDIA; KASS, LAURA; MONCZOR, FEDERICO; RANDI, ANDREA

AhR ligands reactivate LINE-1 retrotransposon in triple-negative breast cancer cells MDA-MB-231 and non-tumorigenic mammary epithelial cells NMuMG

BIOCHEMICAL PHARMACOLOGY; Año: 2020 vol. 175

ECHEVERRÍA, EMILIANA; CABRERA, MAIA; BURGHI, VALERIA; SOSA, MÁXIMO; RIPOLL, SONIA; YANEFF, AGUSTÍN; MONCZOR, FEDERICO; DAVIO, CARLOS; SHAYO, CARINA; FERNÁNDEZ, NATALIA

The Regulator of G Protein Signaling Homologous Domain of G Protein-Coupled Receptor Kinase 2 Mediates Short-Term Desensitization of β3-Adrenergic Receptor

Frontiers in Pharmacology; Año: 2020 vol. 11

BURGHI, VALERIA; ECHEVERRÍA, EMILIANA B.; SOSA, MÁXIMO H.; QUIROGA, DIEGO T.; MUÑOZ, MARINA C.; DAVIO, CARLOS; MONCZOR, FEDERICO; FERNÁNDEZ, NATALIA C.; DOMINICI, FERNANDO P.

Participation of Gαi-Adenylate Cyclase and ERK1/2 in Mas Receptor Signaling Pathways

Frontiers in Pharmacology; Año: 2019 vol. 10

DÍAZ NEBREDA, ANTONELA; ZAPPIA, CARLOS DANIEL; RODRÍGUEZ GONZÁLEZ, ANGELA; SAHORES, ANA; SOSA, MÁXIMO; BURGHI, VALERIA; MONCZOR, FEDERICO; DAVIO, CARLOS; FERNÁNDEZ, NATALIA; SHAYO, CARINA

Involvement of histamine H1 and H2 receptor inverse agonists in receptor's crossregulation

EUROPEAN JOURNAL OF PHARMACOLOGY; Año: 2019 vol. 847 p. 42 - 52

VENTURA, C.; ZAPPIA, C.D.; LASAGNA, M.; PAVICIC, W.; RICHARD, S.; BOLZAN, A.D.; MONCZOR, F.; NÚÑEZ, M.; COCCA, C.

Effects of the pesticide chlorpyrifos on breast cancer disease. Implication of epigenetic mechanisms

JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY; Año: 2019 vol. 186 p. 96 - 104

ZAPPIA, CARLOS D.; MONCZOR, FEDERICO

Therapeutic utility of glucocorticoids and antihistamines cotreatment. Rationale and perspectives

Pharmacology Research & Perspectives; Año: 2019 vol. 7

MONCZOR, FEDERICO; CHATZOPOULOU, ANTONIA; ZAPPIA, CARLOS DANIEL; HOUTMAN, RENÉ; MEIJER, ONNO C.; FITZSIMONS, CARLOS P.

A Model of Glucocorticoid Receptor Interaction With Coregulators Predicts Transcriptional Regulation of Target Genes

Frontiers in Pharmacology; Año: 2019 vol. 10

CAROZZO, ALEJANDRO; YANEFF, AGUSTIN; GOMEZ, NATALIA; DI SIERVI, NICOLAS; SAHORES, ANA; DIEZ, FEDERICO; ATTORRESI, ALEJANDRA I.; RODRIGUEZ-GONZALEZ, ANGELA; MONCZOR, FEDERICO; FERNANDEZ, NATALIA; ABBA, MARTIN; SHAYO, CARINA; DAVIO, CARLOS

IDENTIFICATION OF MRP4/ABCC4 AS A TARGET FOR REDUCING THE PROLIFERATION OF PANCREATIC DUCTAL ADENOCARCINOMA CELLS BY MODULATING THE cAMP EFFLUX

MOLECULAR PHARMACOLOGY; Lugar: Baltimore; Año: 2019

ZAPPIA, CARLOS D.; SOTO, ARIADNA; GRANJA GALEANO, GINA; FENOY, IGNACIO; FERNANDEZ, NATALIA; DAVIO, CARLOS A.; SHAYO, CARINA; FITZSIMONS, CARLOS P.; GOLDMAN, ALEJANDRA; MONCZOR, FEDERICO

Azelastine potentiates antiasthmatic dexamethasone effect on a murine asthma model

Pharmacology Research & Perspectives; Lugar: New York; Año: 2019 vol. 7

GRANJA GALEANO, GINA; ZAPPIA, CARLOS DANIEL; FABIAN, LUCAS; DAVIO, CARLOS; SHAYO, CARINA; FERNANDEZ, NATALIA; MONCZOR, FEDERICO

Effect of mutation of Phe 243 (6.44) of the histamine H 2 receptor on cimetidine and ranitidine mechanism of action

BIOCHEMICAL PHARMACOLOGY; Lugar: Amsterdam; Año: 2017 vol. 146 p. 117 - 126

MONCZOR, FEDERICO; COPSEL, SABRINA; FERNANDEZ, NATALIA; DAVIO, CARLOS; SHAYO, CARINA

Histamine H2 Receptor in Blood Cells: A Suitable Target for the Treatment of Acute Myeloid Leukemia

Handobook of Experimental Pharmacology; Año: 2017

MONCZOR FEDERICO; FERNANDEZ NATALIA

Current Knowledge and Perspectives on Histamine H1 and H2 Receptor Pharmacology: Functional Selectivity, Receptor Crosstalk, and Repositioning of Classic Histaminergic Ligands.

MOLECULAR PHARMACOLOGY; Lugar: Baltimore; Año: 2016 vol. 90 p. 640 - 648

ALONSO NATALIA; DIAZ NEBREDA, ANTONELLA; MONCZOR FEDERICO; GUTKIND SILVIO; DAVIO, CARLOS; FERNANDEZ, NATALIA; SHAYO, CARINA

PI3K pathway is involved in ERK signaling cascade activation by histamine H2R agonist in HEK293T cells.

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS; Lugar: Amsterdam; Año: 2016 vol. 1860 p. 1998 - 2007

ALONSO NATALIA; ZAPPIA, CARLOS DANIEL; CABRERA, MAIA; DAVIO CARLOS; SHAYO CARINA; MONCZOR FEDERICO; FERNANDEZ NATALIA

Physiological implications of biased signaling at histamine H2 receptors.

Frontiers in Pharmacology; Lugar: Lausanne; Año: 2015 vol. 6

ZAPPIA, CARLOS DANIEL; GRANJA GALEANO, GINA; FERNANDEZ NATALIA; SHAYO CARINA; DAVIO CARLOS; FITZSIMONS CARLOS; MONCZOR FEDERICO

Effects of histamine H1 receptor signaling on glucocorticoid receptor activity. Role of canonical and non-canonical pathways.

Scientific Reports; Lugar: London; Año: 2015

ALONSO NATALIA; MONCZOR FEDERICO; ECHEVERRIA, EMILIANA; DAVIO CARLOS; SHAYO CARINA; FERNANDEZ NATALIA

Signal transduction mechanism of biased ligands at histamine H2 receptors.

BIOCHEMICAL JOURNAL; Lugar: Londres; Año: 2014

MONCZOR FEDERICO; FERNANDEZ NATALIA; FITZSIMONS CARLOS; SHAYO CARINA; DAVIO CARLOS

Antihistaminergics and inverse agonism. Potential therapeutic applications.

EUROPEAN JOURNAL OF PHARMACOLOGY; Lugar: Amsterdam; Año: 2013

ALONSO NATALIA; FERNANDEZ NATALIA; NOTCOVICH CINTIA; MONCZOR FEDERICO; SIMAAN MAY; BALDI ALBERTO; GUTKIND SILVIO; DAVIO CARLOS; SHAYO CARINA

Cross-desensitization and cointernalization of h1 and h2 histamine receptors reveal new insights into histamine signal integration.

MOLECULAR PHARMACOLOGY; Lugar: Baltimore; Año: 2013 vol. 83 p. 1087 - 1098

FERNANDEZ NATALIA; GOTTARDO FEDERICO; ALONSO NATALIA; MONCZOR FEDERICO; SHAYO CARINA; DAVIO CARLOS

Roles of phosphorylation-dependent and -independent mechanisms in the regulation of histamine H2 receptor by G protein-coupled receptor kinase 2.

JOURNAL OF BIOLOGICAL CHEMISTRY; Lugar: Bethesda, Maryland; Año: 2011 vol. 286 p. 28697 - 28706

RIVEIRO EUGENIA; DE KIMPE NORBERT; MOGLIONI ALBERTINA; VAZQUEZ RAMIRO; MONCZOR FEDERICO; SHAYO CARINA; DAVIO CARLOS

Coumarins: old compounds with novel promising therapeutic perspectives.

CURRENT MEDICINAL CHEMISTRY.; Año: 2010 vol. 17 p. 1325 - 1338

TUBIO MARIA ROSARIO; FERNANDEZ NATALIA; FITZSIMONS CARLOS; COPSEL SABRINA; SANTIAGO SERGIO DAMIAN; SHAYO CARINA; DAVIO CARLOS; MONCZOR FEDERICO

Expression of a G protein-coupled receptor (GPCR) leads to attenuation of signaling by other GPCRs: experimental evidence for a spontaneous GPCR constitutive inactive form.

JOURNAL OF BIOLOGICAL CHEMISTRY; Año: 2010 vol. 285 p. 14990 - 14998

TAIRA CARLOS; MONCZOR FEDERICO; HÖCHT CHRISTIAN

Measurement of Inverse Agonism in b-Adrenoceptors

METHODS IN ENZYMOLOGY.; Lugar: New York; Año: 2010 vol. 485 p. 37 - 60

FERNANDEZ NATALIA; MONCZOR FEDERICO; BALDI ALBERTO; DAVIO CARLOS; SHAYO CARINA

Histamine H2 receptor trafficking: role of arrestin, dynamin, and clathrin in histamine H2 receptor internalization

MOLECULAR PHARMACOLOGY; Lugar: Bethesda; Año: 2008 vol. 74 p. 1109 - 1118

FERNANDEZ NATALIA; MONCZOR FEDERICO; TUBIO MARIA ROSARIO; SHAYO CARINA; DAVIO CARLOS

Regulatory mechanisms underlying GKR2 levels in U937 cells. Evidence for GRK3 involvement.

BIOCHEMICAL PHARMACOLOGY; Año: 2007 vol. 73 p. 1758 - 1767

MONCZOR FEDERICO; FERNANDEZ NATALIA; RIVEIRO EUGENIA; MLADOVAN ALEJANDRO; BALDI ALBERTO; SHAYO CARINA; DAVIO CARLOS

Histamine H2 receptor overexpression induces U937 cell differentiation despite triggered mechanisms to attenuate cAMP signalling.

BIOCHEMICAL PHARMACOLOGY; Lugar: Amsterdam; Año: 2006 vol. 71 p. 1219 - 1228

MONCZOR FEDERICO

Mechanisms of inverse agonism at histamine H(2) receptors - potential benefits and concerns.

INFLAMMOPHARMACOLOGY; Lugar: Basilea; Año: 2006 vol. 14 p. 89 - 96

FITZSIMONS CARLOS; MONCZOR FEDERICO; FERNANDEZ NATALIA; SHAYO CARINA; DAVIO CARLOS

Mepyramine, a histamine H1 receptor inverse agonist, binds preferentially to a G protein-coupled form of the receptor and sequesters G protein.

JOURNAL OF BIOLOGICAL CHEMISTRY; Año: 2004 vol. 279 p. 34431 - 34439

RIVEIRO EUGENIA; SHAYO CARINA; MONCZOR FEDERICO; FERNANDEZ NATALIA; BALDI ALBERTO; DE KIMPE NORBERT; ROSSI JORGE; DEBENEDETTI SILVIA; DAVIO CARLOS

Induction of cell differentiation in human leukemia U-937 cells by 5-oxygenated-6,7-methylenedioxycoumarins from Pterocaulon polystachyum

CANCER LETTERS; Año: 2004 vol. 210 p. 179 - 188

SHAYO CARINA; LEGNAZZI BL; MONCZOR FEDERICO; FERNANDEZ NATALIA; RIVEIRO EUGENIA; BALDI ALBERTO; DAVIO CARLOS

The time-course of cyclic AMP signaling is critical for leukemia U-937 cell differentiation

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS; Año: 2004 vol. 314 p. 798 - 804

MONCZOR FEDERICO; FERNANDEZ NATALIA; LEGNAZZI BL; RIVEIRO EUGENIA; BALDI ALBERTO; SHAYO CARINA; DAVIO CARLOS

Tiotidine, a histamine H2 receptor inverse agonist that binds with high affinity to an inactive G-protein-coupled form of the receptor. Experimental support for the cubic ternary complex model.

MOLECULAR PHARMACOLOGY; Lugar: New York; Año: 2003 vol. 64 p. 512 - 520

FERNANDEZ NATALIA; MONCZOR FEDERICO; LEGNAZZI BL; NOTCOVICH CINTIA; BALDI ALBERTO; DAVIO CARLOS; SHAYO CARINA

Reduction of G protein-coupled receptor kinase 2 expression in U-937 cells attenuates H2 histamine receptor desensitization and induces cell maturation.

MOLECULAR PHARMACOLOGY; Año: 2002 vol. 62 p. 1506 - 1514

DAVIO CARLOS; MLADOVAN ALEJANDRO; LEGNAZZI BL; MONCZOR FEDERICO; SHAYO CARINA; RIVERA ELENA; BALDI ALBERTO

H1 and H2 histamine receptors mediate the production of inositol phosphates but not cAMP in human breast epithelial cells.

INFLAMMATION RESEARCH; Año: 2002 vol. 51 p. 1 - 7

SHAYO CARINA; FERNANDEZ NATALIA; LEGNAZZI BL; MONCZOR FEDERICO; MLADOVAN ALEJANDRO; BALDI ALBERTO; DAVIO CARLOS

Histamine H2 receptor desensitization: involvement of a select array of G protein-coupled receptor kinases.

MOLECULAR PHARMACOLOGY; Año: 2001 vol. 60 p. 1049 - 1056

LEGNAZZI BL; SHAYO CARINA; MONCZOR FEDERICO; MARTIN MARIA EUGENIA; FERNANDEZ NATALIA; BRODSKY ANDRES; BALDI ALBERTO; DAVIO CARLOS

Rapid desensitization and slow recovery of the cyclic AMP response mediated by histamine H(2) receptors in the U937 cell line.

BIOCHEMICAL PHARMACOLOGY; Año: 2000 vol. 60 p. 159 - 166

MONCZOR FEDERICO; LEGNAZZI BL; RIVERA ELENA; DAVIO CARLOS

Tiotidine, a classical H2-antagonist, presents characteristics of an inverse agonist in U937 cell line.

INFLAMMATION RESEARCH; Lugar: Basilea; Año: 1998 vol. 47 p. 42 - 43

LEGNAZZI BL; MONCZOR FEDERICO; RIVERA ELENA; BERGOC ROSA; DAVIO CARLOS

Histamine receptors in human epithelial cells--characterization of the receptor G-protein-effector system.

INFLAMMATION RESEARCH; Año: 1998 vol. 47 p. 40 - 41