JASINSKI, GABRIEL; SALAS-SARDUY, EMIR; VEGA, DANIEL; FABIAN, LUCAS; FLORENCIA MARTINI, M.; MOGLIONI, ALBERTINA G.

Design, synthesis and biological evaluation of novel thiosemicarbazones as cruzipain inhibitors

EUROPEAN JOURNAL OF MEDICAL CHEMISTRY; Año: 2023 vol. 254

RICCI, ALEJANDRO D.; BRACCO, LEONEL; SALAS-SARDUY, EMIR; RAMSEY, JANINE M.; NOLAN, MELISSA S.; LYNN, M. KATIE; ALTCHEH, JAIME; BALLERING, GRISELDA E.; TORRICO, FAUSTINO; KESPER, NORIVAL; VILLAR, JUAN C.; MARCIPAR, IVÁN S.; MARCO, JORGE D.; AGÜERO, FERNÁN

The Trypanosoma cruzi Antigen and Epitope Atlas: antibody specificities in Chagas disease patients across the Americas

NATURE COMMUNICATIONS; Año: 2023 vol. 14

ANDREA CÓRDOVA ISAZA; SOFÍA JIMÉNEZ MÁRMOL; GUERRA, YASEL; EMIR SALAS SARDUY

Enzyme Inhibitors from Gorgonians and Soft Corals

MARINE DRUGS; Lugar: Basel; Año: 2023 vol. 21 p. 1 - 32

HERNÁNDEZ GONZÁLEZ, JORGE ENRIQUE; SALAS-SARDUY, EMIR; ALVAREZ, LILIAN HERNÁNDEZ; VALIENTE, PEDRO A; ARNI, RAGHUVIR K; PASCUTTI, PEDRO G

Three decades targeting falcipains to develop antiplasmodial agents: what have we learned and what can be done next?

CURRENT MEDICINAL CHEMISTRY.; Año: 2023 vol. 31

GABRIEL JASINSKY; EMIR SALAS SARDUY; DANIEL VEGA; LUCAS FABIAN; MARÍA FLORENCIA MARTINI; MOGLIONI, ALBERTINA G.

Thiosemicarbazone derivatives: evaluation as cruzipain inhibitors and molecular modeling study of complexes with cruzain.

BIOORGANIC & MEDICINAL CHEMISTRY.; Lugar: Amsterdam; Año: 2022

PÉREZ, BRIAN; BOUVIER, LEÓN A.; CAZZULO, JUAN JOSÉ; AGÜERO, FERNÁN; SALAS-SARDUY, EMIR; ALVAREZ, VANINA E.

Screening and identification of metacaspase inhibitors: Evaluation of inhibition mechanism and trypanocidal activity

ANTIMICROBIAL AGENTS AND CHEMOTHERAPY; Año: 2021 vol. 65

HERNÁNDEZ GONZÁLEZ, JORGE ENRIQUE; SALAS-SARDUY, EMIR; HERNÁNDEZ ALVAREZ, LILIAN; BARRETO GOMES, DIEGO ENRY; PASCUTTI, PEDRO GERALDO; OOSTENBRINK, CHRIS; LEITE, VITOR B. P.

In silico identification of noncompetitive inhibitors targeting an uncharacterized allosteric site of falcipain-2

J. COMPUT. AIDED MOL. RESIGN; Año: 2021

HERNÁNDEZ GONZÁLEZ, JORGE ENRIQUE; ALBERCA, LUCAS N.; MASFORROL GONZÁLEZ, YORDANKA; REYES ACOSTA, OSVALDO; TALEVI, ALAN; SALAS-SARDUY, EMIR

Tetracycline Derivatives Inhibit Plasmodial Cysteine Protease Falcipain-2 through Binding to a Distal Allosteric Site

JOURNAL OF CHEMICAL INFORMATION AND MODELING; Lugar: Washington; Año: 2021 vol. 62 p. 159 - 175

SALAS-SARDUY, EMIR; LANDABURU, LIONEL URÁN; CARMONA, ADRIANA K.; CAZZULO, JUAN JOSÉ; AGÜERO, FERNÁN; ALVAREZ, VANINA E.; NIEMIROWICZ, GABRIELA T.

Potent and selective inhibitors for M32 metallocarboxypeptidases identified from high-throughput screening of anti-kinetoplastid chemical boxes

PLoS Neglected Tropical Diseases; Año: 2019 vol. 13

FABIAN, L.; MARTINI, M. FLORENCIA; SARDUY, EMIR SALAS; ESTRIN, DARíO A.; MOGLIONI, ALBERTINA G.

Evaluation of quinoxaline compounds as ligands of a site adjacent to S2 (AS2) of cruzain

BIORGANIC AND MEDICINAL CHEMISTRY LETTERS; Año: 2019 vol. 29 p. 2197 - 2202

SALAS-SARDUY, EMIR; NIEMIROWICZ, GABRIELA T.; JOS� CAZZULO, JUAN; ALVAREZ, VANINA EDER

Target-based screening of the Chagas box: setting up enzymatic assays to discover specific inhibitors across bioactive compounds

CURRENT MEDICINAL CHEMISTRY.; Año: 2019 vol. 26

ALBERCA, LUCAS N.; CHUGURANSKY, SARA R.; ALVAREZ, CORA L.; TALEVI, ALAN; SALAS-SARDUY, EMIR

In silico Guided Drug Repurposing: Discovery of New Competitive and Non-competitive Inhibitors of Falcipain-2

Frontiers in Chemistry; Año: 2019 vol. 7