BARRI, IVAN; RIAFRECHA, LEONARDO E.; ECHEVERRIA, GUSTAVO A.; PIRO, OSCAR A.; COLINAS, PEDRO A.

Spontaneous resolution of diastereomeric glycosyl isoxazolines: A combined theoretical and experimental study in solution and in the crystalline form

JOURNAL OF MOLECULAR STRUCTURE; Lugar: Ámsterdam; Año: 2024 vol. 1310

LE PORS, MACARENA S.; SANTA MARIA DE LA PARRA, LUCÍA; RIAFRECHA, LEONARDO E.; VULLO, DANIELA; LEÓN, IGNACIO E.; SUPURAN, CLAUDIU T.; COLINAS, PEDRO A.

Glycosyl Isoxazoles for Targeting of Tumor Microenvironment and Cancer Cells: Highly Selective Inhibitors of Carbonic Anhydrases IX and XII Showing Cytotoxic Activity

ChemistrySelect; Lugar: Weinheim; Año: 2023 vol. 8

LE PORS, MACARENA S.; BARRI, IVAN; RIAFRECHA, LEONARDO E.; ECHEVERRIA, GUSTAVO A.; PIRO, OSCAR A.; COLINAS, PEDRO ALFONSO

Green Biphasic Synthesis, X‐Ray Diffraction Structure and Conformational Analysis of O ‐Glycosylmethyl Isoxazoles: Potential Substrates of GLUT‐1 Glucose Transporter.

ChemistrySelect; Lugar: Weinheim; Año: 2022 vol. 7

RIAFRECHA, LEONARDO E.; LE PORS, MACARENA S.; LAVECCHIA, MARTÍN J.; BUA, SILVIA; SUPURAN, CLAUDIU T.; COLINAS, PEDRO A.

Vanillin enones as selective inhibitors of the cancer associated carbonic anhydrase isoforms IX and XII. The out of the active site pocket for the design of selective inhibitors?

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY; Año: 2021 vol. 36 p. 2118 - 2127

LLANTÉN MARTÍNEZ, HELBERTH J.; RIAFRECHA, LEONARDO E.; COLINAS, PEDRO A.

C-cinnamoyl Glycosides: An Emerging "Tail" for the Development of Selective Carbonic Anhydrase Inhibitors

CURRENT MEDICINAL CHEMISTRY.; Lugar: Oak Park; Año: 2019 vol. 26 p. 2601 - 2608

RIAFRECHA, LEONARDO E.; BUA, SILVIA; SUPURAN, CLAUDIU T.; COLINAS, PEDRO A.

Improving the carbonic anhydrase inhibition profile of the sulfamoylphenyl pharmacophore by attachment of carbohydrate moieties

BIOORGANIC CHEMISTRY; Lugar: Amsterdam; Año: 2018 vol. 76 p. 61 - 66

ZARO, MARÍA J.; BORTTOLOTI ANA; RIAFRECHA, LEONARDO E.; CONCELLÓN, ANALÍA; MORBIDONI, HÉCTOR R.; COLINAS, PEDRO ALFONSO

Anti-tubercular and antioxidant activities of C-glycosyl carbonic anhydrase inhibitors: towards the development of novel chemotherapeutic agents against Mycobacterium tuberculosis

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY; Lugar: Londres; Año: 2016 vol. 31 p. 1726 - 1730

RIAFRECHA, LEONARDO E.; BUA, SILVIA; SUPURAN, CLAUDIU T.; COLINAS, PEDRO ALFONSO

Synthesis and carbonic anhydrase inhibitory effects of new N-glycosylsulfonamides incorporating the phenol moiety

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS; Lugar: Amsterdam; Año: 2016 vol. 26 p. 3892 - 3895

RIAFRECHA, LEONARDO E.; VULLO, DANIELA; OUAHRANI-BETTACHE, SAFIA; KO¨HLER, STEPHAN; DUMY, PASCAL; WINUM, JEAN-YVES; SUPURAN, CLAUDIU T.; COLINAS, PEDRO ALFONSO

Inhibition of b-carbonic anhydrases from Brucella suis with C-cinnamoyl glycosides incorporating the phenol moiety

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY; Lugar: Londres; Año: 2015 vol. 30 p. 1017 - 1020

RIAFRECHA, LEONARDO E.; VULLO, DANIELA; SUPURAN, CLAUDIU T.; COLINAS, PEDRO ALFONSO

C-glycosides incorporating the 6-methoxy-2-naphthyl moiety are selective inhibitors of fungal and bacterial carbonic anhydrases

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY; Lugar: Londres; Año: 2015 vol. 30 p. 857 - 861

RIAFRECHA, LEONARDO E.; RODRÍGUEZ OSCAR M.; VULLO, DANIELA; SUPURAN, CLAUDIU T.; COLINAS, PEDRO ALFONSO

Attachment of carbohydrates to methoxyaryl moieties leads to highly selective inhibitors of the cancer associated carbonic anhydrase isoforms IX and XII

BIOORGANIC & MEDICINAL CHEMISTRY.; Lugar: Amsterdam; Año: 2014 vol. 22 p. 5308 - 5314

RIAFRECHA, LEONARDO E.; RODRÍGUEZ OSCAR M.; VULLO, DANIELA; SUPURAN, CLAUDIU T.; COLINAS, PEDRO ALFONSO

Synthesis of C-cinnamoyl glycosides and their inhibitory activity against mammalian carbonic anhydrases

BIOORGANIC & MEDICINAL CHEMISTRY.; Lugar: Amsterdam; Año: 2013 vol. 21 p. 1489 - 1494

BUCHIERIE, MARÍA V.; RIAFRECHA, LEONARDO E.; RODRÍGUEZ OSCAR M.; VULLO, DANIELA; MORBIDONI, HÉCTOR R.; SUPURAN, CLAUDIU T.; COLINAS, PEDRO ALFONSO

Inhibition of the b-carbonic anhydrases of Mycobacterium tuberculosis with C-cinnamoyl glycosides: identification of the first inhibitor with antimycobacterial activity

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS; Lugar: Amsterdam; Año: 2013 vol. 23 p. 740 - 743