INVESTIGADORES
COLINAS Pedro Alfonso
artículos
BARRI, IVAN A.; RIAFRECHA, LEONARDO E.; ECHEVERRÍA, GUSTAVO A.; PIRO, OSCAR E.; COLINAS, PEDRO A.
Spontaneous resolution of diastereomeric glycosyl isoxazolines: a combined theoretical and experimental study in solution and in the crystalline form.
JOURNAL OF MOLECULAR STRUCTURE; Año: 2024
LE PORS, MACARENA S.; SANTA MARIA DE LA PARRA, LUCÍA; RIAFRECHA, LEONARDO E.; VULLO, DANIELA; LEÓN, IGNACIO E.; SUPURAN, CLAUDIU T.; COLINAS, PEDRO A.
Glycosyl Isoxazoles for Targeting of Tumor Microenvironment and Cancer Cells: Highly Selective Inhibitors of Carbonic Anhydrases IX and XII Showing Cytotoxic Activity
ChemistrySelect; Lugar: Hoboken; Año: 2023 vol. 8
LE PORS, MACARENA S.; BARRI, IVAN A.; RIAFRECHA, LEONARDO E.; ECHEVERRÍA, GUSTAVO A.; PIRO, OSCAR E.; COLINAS, PEDRO A.
Green Biphasic Synthesis, X‐Ray Diffraction Structure and Conformational Analysis of O ‐Glycosylmethyl Isoxazoles: Potential Substrates of GLUT‐1 Glucose Transporter.
ChemistrySelect; Lugar: Hoboken; Año: 2022 vol. 7
RIAFRECHA, LEONARDO E.; LE PORS, MACARENA S.; LAVECCHIA, MARTÍN, J.; BUA, SILVIA; SUPURAN, CLAUDIU T.; COLINAS, PEDRO ALFONSO
Vanillin enones as selective inhibitors of the cancer associated carbonic anhydrase isoforms IX and XII. The out of the active site pocket for the design of selective inhibitors?
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY; Lugar: Londres; Año: 2021 vol. 36 p. 2118 - 2127
LLANTÉN MARTÍNEZ, HELBERTH J.; RIAFRECHA, LEONARDO E.; COLINAS, PEDRO ALFONSO
C-cinnamoyl Glycosides: An Emerging ?Tail? for the Development of Selective Carbonic Anhydrase Inhibitors
CURRENT MEDICINAL CHEMISTRY.; Lugar: Oak Park; Año: 2019 vol. 26 p. 2601 - 2608
RIAFRECHA, LEONARDO E.; BUA, SILVIA; SUPURAN, CLAUDIU T.; COLINAS, PEDRO A.
Improving the carbonic anhydrase inhibition profile of the sulfamoylphenyl pharmacophore by attachment of carbohydrate moieties
BIOORGANIC CHEMISTRY; Año: 2018 vol. 76 p. 61 - 66
LLANTÉN MARTÍNEZ, HELBERTH J.; BARATA, S.; POSTIGO, A.; COLINAS, PEDRO ALFONSO
Synthesis of C-glycosylmethyl isoxazoles via aerobic oxidation of ketoximes catalyzed by TEMPO
TETRAHEDRON LETTERS; Lugar: Amsterdam; Año: 2017 vol. 58 p. 1507 - 1511
RIAFRECHA, LEONARDO E.; BUA, SILVIA; SUPURAN, CLAUDIU T.; COLINAS, PEDRO ALFONSO
Synthesis and carbonic anhydrase inhibitory effects of new N-glycosylsulfonamides incorporating the phenol moiety
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS; Lugar: Amsterdam; Año: 2016 vol. 26 p. 3892 - 3895
AZARO, MARÍA JOSE; BORTOLOTTI, ANA; RIAFRECHA, LEONARDO E.; CONCELLÓN, ANALÍA; MORBIDONI, HÉCTOR R.; COLINAS, PEDRO ALFONSO
Anti-tubercular and antioxidant activities of C-glycosyl carbonic anhydrase inhibitors: Towards the development of novel chemotherapeutic agents against Mycobacterium tuberculosis
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY; Lugar: Londres; Año: 2016 vol. 31 p. 1726 - 1730
RIAFRECHA, LEONARDO E.; VULLO, DANIELA; OUAHRANI-BETTACHE, SAFIA ; KÖHLER, STEPHAN; DUMY, PASCAL; WINUM, JEAN-YVES; SUPURAN, CLAUDIU T.; COLINAS PEDRO ALFONSO
Inhibition of betha-carbonic anhydrases from Brucella suis with C-cinnamoyl glycosides incorporating the phenol moiety
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY; Lugar: Londres; Año: 2015 vol. 30 p. 1017 - 1020
RIAFRECHA, LEONARDO E.; VULLO, DANIELA; SUPURAN, CLAUDIU T.; COLINAS, PEDRO ALFONSO
C-glycosides incorporating the 6-methoxy-2-naphthyl moiety are selective inhibitors of fungal and bacterial carbonic anhydrases
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY; Lugar: Londres; Año: 2015 vol. 30 p. 857 - 861
RIAFRECHA, LEONARDO E.; RODRÍGUEZ OSCAR M.; VULLO, DANIELA; SUPURAN, CLAUDIU T.; COLINAS, PEDRO ALFONSO
Attachment of carbohydrates to methoxyaryl moieties leads to highly selective inhibitors of the cancer associated carbonic anhydrase isoforms IX and XII
BIOORGANIC & MEDICINAL CHEMISTRY.; Lugar: Amsterdam; Año: 2014 vol. 22 p. 5308 - 5314
RIAFRECHA, LEONARDO E.; RODRÍGUEZ OSCAR M.; VULLO, DANIELA; SUPURAN, CLAUDIU T.; COLINAS, PEDRO ALFONSO
Synthesis of C-cinnamoyl glycosides and their inhibitory activity against mammalian carbonic anhydrases
BIOORGANIC & MEDICINAL CHEMISTRY.; Lugar: Amsterdam; Año: 2013 vol. 21 p. 1489 - 1494
COLINAS PEDRO ALFONSO
Novel sulfonamide compounds for inhibition of metastatic tumor growth (WO2012021963)
EXPERT OPINION ON THERAPEUTIC PATENTS; Lugar: London; Año: 2013 vol. 23 p. 761 - 763
WINUM, JEAN-YVES; COLINAS, PEDRO ALFONSO; SUPURAN, CLAUDIU T.
Glycosidic Carbonic Anhydrase IX Inhibitors: a Sweet Approach against Cancer.
BIOORGANIC & MEDICINAL CHEMISTRY.; Lugar: Amsterdam; Año: 2013 vol. 21 p. 1419 - 1426
BUCHIERI, MARÍA V; RIAFRECHA, LEONARDO E.; RODRÍGUEZ OSCAR M.; VULLO, DANIELA; MORBIDONI, HÉCTOR R.; SUPURAN, CLAUDIU T.; COLINAS, PEDRO ALFONSO
Inhibition of the b-carbonic anhydrases of Mycobacterium tuberculosis with C-cinnamoyl glycosides: identification of the first inhibitor with antimycobacterial activity
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS; Lugar: Amsterdam; Año: 2013 vol. 23 p. 740 - 743
CAMÍ, GERARDO; CHACÓN VILLALBA, E.; COLINAS, PEDRO ALFONSO; ECHEVERRÍA, GUSTAVO; ESTIÚ, G.; SORIA, DELIA B.
Crystal structure, Spectroscopy and theoretical studies of p-cyanobenzenosulfonamide and a Cu(II) complex
JOURNAL OF MOLECULAR STRUCTURE; Lugar: Amsterdam; Año: 2012 vol. 1024 p. 110 - 116
LAVECCHIA, MARTÍN, J.; RODRÍGUEZ OSCAR M.; ECHEVERRÍA, GUSTAVO; PIS DIEZ, REYNALDO; COLINAS, PEDRO ALFONSO
Conformational behavior of peracetylated b-D-mannopyranosyl methanesulfonamide: implications for the mechanism of sulfonamidoglycosylation of carbohydrate derivatives.
CARBOHYDRATE RESEARCH; Lugar: Amsterdam; Año: 2012 vol. 361 p. 182 - 188
COLINAS PEDRO ALFONSO
Novel Glycomimetics: Anomeric and N-Glycosyl Sulfonamides
CURRENT ORGANIC CHEMISTRY; Lugar: Oak Park; Año: 2012 vol. 16 p. 1670 - 1679
LAVECCHIA, MARTÍN, J.; PIS DIEZ, REYNALDO; COLINAS, PEDRO ALFONSO
A combined theoretical and spectroscopic study of 4,6-di-O-acetyl-2,3-dideoxy-D-erythro-hex-2-enopyranosyl sulfamide: a novel glycosyl carbonic anhydrase IX inhibitor
CARBOHYDRATE RESEARCH; Año: 2011 vol. 346 p. 435 - 441
CAMÍ, GERARDO; CHACÓN VILLALBA, E.; DI SANTI, Y.; COLINAS PEDRO ALFONSO; ESTIÚ, G.; SORIA, DELIA B.
Synthesis, Thermogravimetric, Spectroscopic and Theoretical Characterization of copper(II) complex with 4-chloro-2-nitrobenzenosulphonamide.
JOURNAL OF MOLECULAR STRUCTURE; Año: 2011 vol. 995 p. 72 - 77
RODRÍGUEZ OSCAR M.; MARESCA ALFONSO; TÉMPERA, CARLOS AGUSTÍN; BRAVO, R. D.; COLINAS, PEDRO ALFONSO; SUPURAN, CLAUDIU T.
N-b-glycosyl sulfamides are selective inhibitors of the cancer associated carbonic anhydrase isoforms IX and XII
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS; Año: 2011 vol. 21 p. 4447 - 4450
CRESPO, ROSANA; BRAVO, MARGARITA G. DE; COLINAS, PEDRO ALFONSO; BRAVO, RODOLFO D.
In vitro antitumor activity of N-glycosyl sulfonamides
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS; Año: 2010 vol. 20 p. 6469 - 6471
TÉMPERA, CARLOS AGUSTÍN; COLINAS, PEDRO ALFONSO; BRAVO RODOLFO D.
Efficient synthesis of 2,3-unsaturated sulfonamidoglycosides by Amberlyst 15
TETRAHEDRON LETTERS; Año: 2010 vol. 51 p. 5372 - 5374
COLINAS PEDRO ALFONSO; TÉMPERA, CARLOS AGUSTÍN; RODRÍGUEZ OSCAR M.; BRAVO, RODOLFO DANIEL
Stereoselective synthesis of new N-betha-glycosyl sulfonamides by sulfonamidoglycosylation of per-O-acetylated sugars
SYNTHESIS-STUTTGART; Lugar: Stuttgart; Año: 2009 vol. 2009 p. 4143 - 4148
ALEGRE, MARÍA LUJÁN; PIS DIEZ, REYNALDO; COLINAS PEDRO ALFONSO
Experimental and theoretical study of the conformational, vibrational and magnetic properties of 4,6-di-O-acetyl-2,3-dideoxy-D-threo-hex-2-enopyranosyl ethanesulfonamide
JOURNAL OF MOLECULAR STRUCTURE; Año: 2009 vol. 919 p. 223 - 226
VEGA ENRIQUE D.; COLINAS, PEDRO ALFONSO
ADSORPTION OF FUMARIC AND MALEIC ACIDS ONTO HYDROXYAPATITE: A THERMODYNAMIC STUDY
Journal of the Argentine Chemical Society; Lugar: Buenos Aires; Año: 2009 vol. 97 p. 195 - 206
RODRÍGUEZ OSCAR M.; COLINAS PEDRO ALFONSO; BRAVO RODOLFO D.
Synthesis of 2,3-unsaturated O- and N-glycosides by HBF4.SiO2 catalyzed
SYNLETT; Año: 2009 vol. 7 p. 1154 - 1156
COLINAS, PEDRO ALFONSO; NUÑEZ, NICOLÁS ANTONIO; BRAVO, RODOLFO DANIEL
Sulfonamidoglycosylation of methyl glycosides employing perchloric acid supported on silica gel
JOURNAL OF CARBOHYDRATE CHEMISTRY; Año: 2008 vol. 27 p. 141 - 147
COLINAS, PEDRO ALFONSO; BRAVO, RODOLFO DANIEL; ECHEVERRÍA GUSTAVO
X-ray crystallographic and high-resolution NMR spectroscopy characterization of 4,6-di-O-acetyl-2,3-dideoxy-alpha-D-erytrho-hex-2-enopyranosyl sulfamide
CARBOHYDRATE RESEARCH; Año: 2008 vol. 343 p. 3005 - 3008
COLINAS, PEDRO ALFONSO; BRAVO, RODOLFO DANIEL
Ferrier sulfonamidoglycosylation of D-glycals
CARBOHYDRATE RESEARCH; Año: 2007 vol. 342 p. 2297 - 2302
COLINAS, PEDRO ALFONSO; BRAVO, RODOLFO DANIEL; VULLO, DANIELA; SCOZZAFAVA, ANDREA; SUPURAN, CLAUDIU T.
Carbonic anhydrase inhibitors. Inhibition of cytosolic isoforms I and II, and extracellular isoforms IV, IX, and XII with sulfamides incorporating sugar moieties
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS; Año: 2007 vol. 17 p. 5086 - 5090
PONZINIBBIO AGUSTÍN; COLINAS PEDRO A.; LIEBERKNECHT ALBRECHT; BRAVO RODOLFO D.
An efficient and stereoselective synthesis of 2-deoxy ketopyranoses from exo-glycals
Letters in Organic Chemistry; Año: 2006 vol. 3 p. 459 - 462
COLINAS PEDRO A.; BRAVO RODOLFO D.
Sulfonamidoglycosylation of methyl ribofuranosides: a novel approach to furanosylsulfonamides
TETRAHEDRON LETTERS; Año: 2005 vol. 46 p. 1687 - 1689
COLINAS PEDRO A.; BRAVO RODOLFO D.
A novel sulfonamidoglycosylation of glycals
ORGANIC LETTERS; Año: 2003 vol. 5 p. 4509 - 4511
COLINAS PEDRO A.; PONZINIBBIO AGUSTÍN; LIEBERKNECHT ALBRECHT; BRAVO RODOLFO D.
Wittig reaction of glycosyl phosphonium salts: a stereoselective route to C-disaccharides and C,O-trisaccharides
TETRAHEDRON LETTERS; Año: 2003 vol. 44 p. 7985 - 7988
COLINAS PEDRO A.; JAEGER VOLKER; LIEBERKNECHT ALBRECHT; BRAVO RODOLFO D.
Nitrile oxide cycloadditions to olefinated sugars
TETRAHEDRON LETTERS; Año: 2003 vol. 44 p. 1071 - 1074
COLINAS PEDRO A.; LIEBERKNECHT ALBRECHT; BRAVO RODOLFO D.
Stereoselective glycosidations of olefinated sugars
TETRAHEDRON LETTERS; Año: 2002 vol. 43 p. 9065 - 9068
LIEBERKNECHT ALBRECHT; GRIESSER, HELMUT; KRAEMER, BERND; BRAVO, RODOLFO D.; COLINAS, PEDRO ALFONSO; GRIGERA, RAÚL J.
Diastereoselective synthesis of -(3,4,6-Tri-O-benzyl-2-deoxy-b-D-lyxo-hexopyranosyl)-N-tert-butoxycarbonyl-D-alanine
TETRAHEDRON; Lugar: Amsterdam; Año: 1999 vol. 55 p. 6475 - 6482
LIEBERKNECHT, ALBRECHT; GRIESSER, HELMUT; BRAVO, RODOLFO D.; COLINAS, PEDRO ALFONSO; GRIGERA, RAÚL J.
Stereoselective Synthesis of Olefinated Sugars
TETRAHEDRON; Lugar: Amsterdam; Año: 1998 vol. 54 p. 3159 - 3168
FREY, WOLFGANG; LIEBERKNECHT, ALBRECHT; GRIESSER, HELMUT; BRAVO, RODOLFO D.; COLINAS, PEDRO ALFONSO; GRIGERA, RAÚL J.
Crystal Structure of (2S, 4R, 5R, 6R)-2-(4,5-Dibenzyloxymethyltetrahydropyranyl) triphenylphosphonium tetrafluorborate, -C45H44PBF4O4 and of (2R, 4R, 5R, 6R)-2-(4,5-Dibenzyloxymethyltetrahydropyranyl) triphenylphosphonium tetrafluorborate, -C45H44PBF4O4
ZEITSCHRIFT FUR KRISTALLOGRAPHIE-NEW CRYSTAL STRUCTURES; Lugar: Munich; Año: 1998 vol. 213 p. 737 - 740
FREY, WOLFGANG; LIEBERKNECHT ALBRECHT; GRIESSER, HELMUT; BRAVO, RODOLFO D.; COLINAS, PEDRO ALFONSO; GRIGERA, RAÚL J.
Crystal Structure of (2R, 4S, 5R)-2-(4-Benzyloxy-5-benzyloxymethyltetrahydrofuranyl)
ZEITSCHRIFT FUR KRISTALLOGRAPHIE-NEW CRYSTAL STRUCTURES; Lugar: Munich; Año: 1998 vol. 213 p. 365 - 366
FREY, WOLFGANG; LIEBERKNECHT, ALBRECHT; GRIESSER, HELMUT; BRAVO, RODOLFO D.; COLINAS, PEDRO ALFONSO; GRIGERA, RAÚL J.
Crystal Structure of (E)-2,5-Anhydro-3-deoxy-4,6-di-O-benzyl-1-p-methoxyphenyl-D-
ZEITSCHRIFT FUR KRISTALLOGRAPHIE-NEW CRYSTAL STRUCTURES; Lugar: Munich; Año: 1998 vol. 213 p. 75 - 76
FREY, W.; LIEBERKNECHT, A.; GRIESSER, H.; BRAVO, R.D.; COLINAS, P.A.; GRIGERA, R.J.
Crystal structure of (2R,4S,5R)-2-(4-benzyloxy-5-benzyloxymethyltetrahydrofuranyl)triphenylphosphonium tetrafluoroborate tetrachloromethane solvate, C37H36PBF4O3 · CCI4
ZEITSCHRIFT FUR KRISTALLOGRAPHIE-NEW CRYSTAL STRUCTURES; Año: 1998 vol. 213 p. 379 - 380
FREY, W.; LIEBERKNECHT, A.; GRIESSER, H.; BRAVO, R.D.; COLINAS, P.A.; GRIGERA, R.J.
Crystal structure of (2R,4S,5R)-2-(4-benzyloxy-5-benzyloxymethyltetrahydrofuranyl)triphenylphosphonium tetrafluoroborate tetrachloromethane solvate, C37H36PBF4O3 · CCI4
ZEITSCHRIFT FUR KRISTALLOGRAPHIE-NEW CRYSTAL STRUCTURES; Año: 1998 vol. 213 p. 379 - 380