INVESTIGADORES
ENRIZ Ricardo Daniel
artículos
Título:
Synthesis of 3-amino-2-ethoxycarbonyl Pyrido [1,2-a]Thieno-[2,3-d]-4-pyrimidone derivatives and their antimalarial and Cytotoxic activities in vitro
Autor/es:
J.CHARRIS; J.DOMINGUEZ; M.CORDERO; L.ORFILA; F.RIGGIONE; S.LOPEZ; ENRIZ R D; F.SUVIRE
Revista:
HETEROCYCLIC COMMUNICATIONS
Editorial:
FREUND PUBLISHING HOUSE LTD
Referencias:
Año: 2000 vol. 6 p. 571 - 578
ISSN:
0793-0283
Resumen:
a series of 3-amino-2-amino-ethoxycarbonylpyrido1,2,a)thieno(2,3-d)-4-pyrimidine 10-13 were prepared in order to investigate their cytotoxicity and antimalarial activities. Some of them showed a promising activities. The detailes synthesis, spectroscopic, computational and biological data are described.